Cyproterone
About Cyproterone
Cyproterone is a prescription hormone treatment primarily used to manage advanced prostate cancer in men. It is also used in women to treat severe symptoms caused by high levels of male sex hormones, such as excessive hair growth and severe acne. This medicine works by blocking hormones that can cause these conditions to worsen.
You must take this medicine consistently at the same times every day as directed by your doctor. It is usually best to take Cyproterone after eating a meal to help prevent stomach upset and ensure proper absorption. Along with this medication, eating a balanced diet, staying hydrated, and avoiding smoking can support your body's response to the treatment.
While taking Cyproterone, you may experience mild side effects like fatigue, weight fluctuations, or mild mood shifts. However, you should contact your doctor immediately if you experience serious symptoms such as yellowing of your skin or eyes, severe abdominal pain, or sudden breathing difficulties.
Before you begin taking this medication, tell your doctor if you have diabetes, blood clotting issues, or chronic depression. Do not take this if you have active liver disease, a history of benign brain tumours, or severe wasting diseases. It is crucial to ensure this medicine is safe for your specific health background.
This medication can interact with certain anti-fungal drugs, seizure medicines, and alcohol, which can strain your liver or make the treatment less effective. Special care and medical advice are needed if you are elderly, and you must never take this if you are pregnant or breastfeeding. Always check with your healthcare team before starting any new treatments or supplements.
Uses of Cyproterone
Medicinal Benefits
Cyproterone helps manage conditions caused by hormone imbalance or hormone-sensitive diseases by reducing the effects of certain hormones in the body. It can improve symptoms and support long-term disease control when used as prescribed.
- Helps Control Hormone-Sensitive Conditions: In conditions such as advanced prostate cancer, Cyproterone helps reduce the effects of male hormones, which can help slow disease progression and relieve associated symptoms.
- Relieves Symptoms of Excess Androgens: In women with conditions related to high androgen levels, Cyproterone may help reduce acne and excessive hair growth, supporting healthier skin and improved comfort.
- Improves Daily Wellbeing: By reducing hormone-related symptoms, Cyproterone can help improve physical comfort, confidence, and quality of life during long-term treatment.
Directions for Use
- Take Cyproterone with food to enhance its absorption.
- Follow your doctor’s instructions on the dosage and timing of this medication, to ensure the safety.
- Swallow the medicine as a whole with a glass of water.
- Do not crush, break, or chew it.
Storage
Side Effects of Cyproterone
Common Side Effects (Usually mild):
- Feeling unusually tired or weak
- Changes in body weight (gain or loss)
- Decreased sex drive or temporary inability to get an erection
- Breast swelling or tenderness
Serious Side Effects (Consult a doctor right away):
- Yellowing of the skin or eyes, dark urine, or severe upper stomach pain (signs of liver damage)
- Sudden shortness of breath, sharp chest pain, or swelling and warmth in one of your legs (signs of blood clots)
- Severe depression, sudden anxiety, or extreme mood changes
- Unusual shortness of breath, dry cough, or persistent breathing issues
- Changes in your vision, severe headaches, or loss of balance
Medicines Containing this Salt
View AllDrug Warnings
- Keep all appointments for regular blood tests so your doctor can monitor your liver function and blood counts.
- Be alert for signs of blood clots, and seek immediate medical help if you notice swelling in one calf, sudden chest pain, or difficulty breathing.
- Do not drive, ride a bicycle, or operate heavy machinery if you feel dizzy, exhausted, or physically weak after taking your dose.
- Tell any doctor, dentist, or surgeon treating you that you are taking Cyproterone, especially if you are planning to have surgery.
- Report any new or worsening headaches, changes in your hearing, or visual disturbances to your doctor right away.
Drug Interactions
- Anti-fungal medications (such as ketoconazole): May increase the concentration of Cyproterone in your blood, raising the risk of side effects.
- Seizure medicines (such as phenytoin or carbamazepine): May speed up how your body breaks down Cyproterone, making it less effective.
- Diabetes medications (including insulin): Cyproterone may affect your blood sugar levels, meaning your doctor might need to adjust your diabetes treatment.
Drug-Drug Interactions Checker List:
Safety Advice
Alcohol
cautionAvoid alcohol consumption while on treatment with Cyproterone.
Pregnancy
unsafeCyproterone is only for use in men. Women should not take this medication.
Breast Feeding
cautionCyproterone is only for use in men. Women should not take this medication.
Driving
cautionCyproterone may affect your reactions and your ability to drive. Do not drive and/or operate machines that require your alertness.
Liver
cautionInform your doctor if you have liver disease. It is not advised to use if you have a history of liver disease (including previous or existing liver tumours (unless caused by secondary cancers caused by prostate cancer), Dubin-Johnson Syndrome, or Rotor Syndrome).
Kidney
cautionInform your doctor before using Cyproterone if you have a kidney impairment/disorder history. Your doctor will prescribe only if the benefits outweigh the risks.
Children
cautionThe safety and effectiveness of Cyproterone in pediatric patients have not been established.
Habit Forming
Diet & Lifestyle Advise
- Support your liver health: Since this medicine is processed by the liver, avoid drinking alcohol entirely, as it increases the risk of severe liver strain.
- Protect your bones: Long-term use of hormone-blocking therapies can weaken bones. Ensure you get enough calcium and vitamin D through foods like leafy greens, fortified dairy, or supplements if recommended by your doctor.
- Stay active: Engage in regular, low-impact exercise like walking or light strength training to combat fatigue and help maintain muscle mass.
- Monitor blood sugar: If you have diabetes, check your blood sugar levels more frequently, as hormone treatments can affect how your body manages glucose.
Special Advise
- Cyproterone should be taken under strict medical supervision. The doctor will regularly monitor your condition while taking Cyproterone.
- Your doctor may get routine blood tests done to monitor your liver function, electrolyte levels, and blood cell count in your blood.
- Peripheral blood counts should be frequently monitored during Cyproterone treatment and, when appropriate, until recovery is achieved.
- Do not donate sperm during treatment with Cyproterone for three months after your last dose.
- If you have diabetes, your doctor may need to alter the dose of medicine required to treat your diabetes.
Patients Concern
Disease/Condition Glossary
Cancer: Cancer is a condition where cells in a specific body part grow and reproduce uncontrollably. The cancerous cells can invade and destroy surrounding healthy tissue, including organs. Cancer sometimes begins in one body part before spreading to other areas.
Prostate cancer: Prostate cancer is a type of cancer that only occurs in men and affects the prostate gland, a tiny gland under the bladder that produces semen. Inability to urinate easily, pain, numbness, or sexual issues are among the symptoms. For men, it is the most typical type of cancer. Although the exact cause of prostate cancer is unknown, it may be brought on by family history, chemical exposure, or both. Prostate cancer risk factors include a family history of the disease, advanced age, obesity, and genetic changes.
FAQs
Cyproterone is used to treat Prostate Cancer.
Most prostate cancers require testosterone to grow. Cyproterone contains Cyproterone, which blocks testosterone, a hormone, from reaching prostate cancer cells. Thus, Cyproterone can slow the cancer's growth and cause it to shrink.
Cyproterone is generally intended for use in men with prostate cancer and should not be used by women unless specifically prescribed for another medical condition. Women who are pregnant or breastfeeding should not take Cyproterone because it may harm an unborn baby or nursing infant. Consult a doctor before any use.
Yes, Cyproterone was generally a well-tolerated medication. Take Cyproterone pills exactly as directed by your healthcare provider. Do not change your dose or stop taking Cyproterone unless your healthcare physician instructs you. If you encounter side symptoms, your healthcare provider may temporarily discontinue your Cyproterone therapy or adjust your Cyproterone dose.
In some cases, Cyproterone may cause decreased fertility in men. However, you should not assume that your female partner cannot become pregnant. Please discuss with your doctor if you have any concerns.
Yes, Cyproterone can cause liver problems, including severe liver damage. Your doctor will perform regular blood tests to check how well your liver is working while you are on this medicine. If you notice yellowing of your skin or eyes, contact your doctor immediately. Talk to your doctor.
You should swallow the tablet whole with water, preferably after a meal. Do not crush, chew, or break the tablet, as this can affect how the medicine is absorbed. Talk to your doctor.
Yes, this medicine can cause drowsiness, fatigue, or dizziness, especially when you first start taking it. Avoid driving or operating machinery until you know how it affects you. Talk to your doctor.
Take the missed dose as soon as you remember, unless it is nearly time for your next dose. Do not take a double dose to make up for a missed tablet. Talk to your doctor.
Yes, mood swings, depressive moods, and severe depression are known side effects of this medicine. If you experience persistent sadness or severe emotional changes, seek medical advice right away. Talk to your doctor.
No, you should avoid alcohol while on this medication. Alcohol can increase the risk of liver strain and make side effects like fatigue much worse. Talk to your doctor.
No, Cyproterone is not typically used to treat male pattern baldness, as its strong hormone-blocking properties can cause unwanted side effects in men. It is sometimes used for women with hair loss related to high androgen levels. Talk to your doctor.

